Telaglenastat
| Catalog Number | Pack Size | List Price* | Quantity | |
|---|---|---|---|---|
| HY-12248-5MG | 5 mg | 89,00 | Add | |
| HY-12248-1ML | 10mM/1mL | 109,00 | Add | |
| HY-12248-10MG | 10 mg | 128,00 | Add | |
| HY-12248-50MG | 50 mg | 356,00 | Add | |
| HY-12248-100MG | 100 mg | 584,00 | Add | |
| HY-12248-500MG | 500 mg | 1'723,00 | Add | |
| HY-12248-S-1ST | Sample | Inquire |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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Telaglenastat (CB-839) is a first-in-class, selective, reversible and orally active glutaminase 1 (GLS1) inhibitor. Telaglenastat selectively inhibits GLS1 splice variants KGA (kidney-type glutaminase) and GAC (glutaminase C) compared to GLS2. The IC50s are 23 nM and 28 nM for endogenous glutaminase in mouse kidney and brain, respectively. Telaglenastat inuduces autophagy and has antitumor activity[1].
| Category | Biochemicals |
| Supplier | MedChem Express |
| Regulatory Status | RUO |
| Research Field | Cancer, Autophagy,Metabolic Enzyme/Protease |
| Format | Solubility: DMSO : 50 mg/mL (ultrasonic) |
| Grade | Clinical information: Phase 2 |
| Purity | 99.92% |
| Molecular Formula | C26H24F3N7O3S |
| Molecular Weight | 571.57 |
| CAS-Number | 1439399-58-2 |
| Storage Conditions | -20°C, 3 years; 4°C, 2 years (Powder) |
| Tech. Data Sheet | View datasheet |
| Link To Supplier | http://www.medchemexpress.com |
| Shipping Details | Room Temperature |
| Material Safety Data Sheet | Download PDF |
