Androgen receptor antagonist 1
| Catalog Number | Pack Size | List Price* | Quantity | |
|---|---|---|---|---|
| HY-130992-5MG | 5 mg | 584,00 | Add | |
| HY-130992-1ML | 10mM/1mL | 641,00 | Add | |
| HY-130992-10MG | 10 mg | 1'027,00 | Add | |
| HY-130992-25MG | 25 mg | 1'977,00 | Add | |
| HY-130992-50MG | 50 mg | 2'990,00 | Add |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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Androgen receptor antagonist 1 is an orally available full androgen receptor (AR) antagonist with an IC50 of 59 nM[1]. Androgen receptor antagonist 1 (Compound 6) can be used in the synthesis of PROTAC AR degraders, which results 24% and 47 % AR protein degradation in LNCaP cells at 1 μM and 10 μM, respectively[2].
| Category | Protein |
| Supplier | MedChem Express |
| Regulatory Status | RUO |
| Research Field | Cancer, PROTAC,Vitamin D Related/Nuclear Receptor |
| Format | Solubility: DMSO : 100 mg/mL (ultrasonic) |
| Grade | Clinical information: No Development Reported |
| Purity | 99.71% |
| Molecular Formula | C21H25ClN4O3 |
| Molecular Weight | 416.9 |
| CAS-Number | 1338812-36-4 |
| Storage Conditions | -20°C, 3 years; 4°C, 2 years (Powder) |
| Tech. Data Sheet | View datasheet |
| Link To Supplier | http://www.medchemexpress.com |
| Shipping Details | Room Temperature |
| Material Safety Data Sheet | Download PDF |
