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CP-100356 hydrochloride


Catalog Number Pack Size List Price* Promo Price* Quantity
HY-108347-5MG 5 mg 537,00 456,50 Add

* CHF, excl. 7.7% VAT and shipping costs


Product Description

CP-100356 hydrochloride is an orally active dual MDR1/BCRP inhibitor, with an IC50s of 0.5 and 1.5 µM for inhibiting MDR1-mediated Calcein-AM transport and BCRP-mediated Prazosin transport, respectively. CP-100356 hydrochloride is also a weak inhibitor of OATP1B1 (IC50=∼66 µM). CP-100356 hydrochloride is devoid of MRP2 and major human P450 enzymes inhibition (IC50>15 µM).

Category Biochemicals
Supplier MedChem Express
Application Metabolism-protein/nucleotide metabolism
Regulatory Status RUO
Grade Clinical information: No Development Reported
Molecular Formula C31H37ClN4O6
Molecular Weight 597.1
CAS-Number [142715-48-8]
Storage Conditions Powder -20°C 3 years, 4°C 2 years; In solvent -80°C 6 months, -20°C 1 month
Product Line Research
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Material Safety Data Sheet Download PDF
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