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PF-06843195


Catalog Number Pack Size List Price* Quantity
HY-131972-50MG 50 mg Inquire
HY-131972-5MG 5 mg Inquire
HY-131972-25MG 25 mg Inquire
HY-131972-10MG 10 mg Inquire
HY-131972-100MG 100 mg Inquire

* CHF, excl. 7.7% VAT and shipping costs


Product Description

PF-06843195 is a highly selective PI3Kα inhibitor with an IC50 of 18 nM in Rat1 fibroblasts. The Kis of PF-06843195 for PI3Kα and PI3Kδ in biochemical kinase assay are less than 0.018 nM and 0.28 nM, respectively. PF-06843195 has great suppression of the PI3K/mTOR signaling pathway and durable antitumor efficacy.

Category Biochemicals
Supplier MedChem Express
Application Cancer-Kinase/protease
Regulatory Status RUO
Grade Clinical information: No Development Reported
Molecular Formula C20H25F3N8O4
Molecular Weight 498.46
CAS-Number [2067281-51-8]
Storage Conditions Please store the product under the recommended conditions in the Certificate of Analysis.
Product Line Research
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Material Safety Data Sheet Download PDF
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