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Article Status


nAChR agonist 1


Catalog Number Pack Size List Price* Promo Price* Quantity
HY-133011-5MG 5 mg 537,00 456,50 Add
HY-133011-10MMO 10 mM * 1 mL 591,00 502,40 Add
HY-133011-10MG 10 mg 881,00 748,90 Add
HY-133011-25MG 25 mg 1'814,00 1'541,90 Add
HY-133011-50MG 50 mg 2'803,00 2'382,60 Add

* CHF, excl. 7.7% VAT and shipping costs


Product Description

nAChR agonist 1 is a potent, brain-permeable, and orally efficacious positive allosteric modulator of α7 nicotinic acetylcholine receptor (α7 nAChR). nAChR agonist 1 has the EC50 of 0.32 µM in a Ca2+ mobilization assay (PNU-282987-induced, FLIPR based) in human IMR-32 neuroblastoma cells that endogenously express α7 nAChR. nAChR agonist 1 can be develpoped for the treatment of Alzheimer’s disease.

Category Biochemicals
Supplier MedChem Express
Application Neuroscience-Neurodegeneration
Regulatory Status RUO
Format Solubility: DMSO : 125 mg/mL (297.66 mM; Need ultrasonic)
Grade Clinical information: Phase 1
Molecular Formula C20H18ClNO3S2
Molecular Weight 419.94
CAS-Number [1394371-75-5]
Storage Conditions Please store the product under the recommended conditions in the Certificate of Analysis.
Product Line Research
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Material Safety Data Sheet Download PDF
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