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Catalog Number Pack Size List Price* Quantity
HY-133016-5MG 5 mg Inquire
HY-133016-25MG 25 mg Inquire
HY-133016-10MG 10 mg Inquire
HY-133016-50MG 50 mg Inquire
HY-133016-100MG 100 mg Inquire

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Product Description

M8891 is an orally active, reversible and brain penetrant Methionine Aminopeptidase-2 (MetAP-2) inhibitor with an IC50 of 54 nM and a Ki of 4.33 nM. M8891 does not inhibit MetAP-1 (IC50>10 µM). M8891 inhibits growth of primary endothelial cells as well as tumor cells and demonstrates antiangiogenic and antitumoral activity.

Category Biochemicals
Supplier MedChem Express
Application Cancer-programmed cell death
Regulatory Status RUO
Format Solubility: DMSO : 125 mg/mL (324.37 mM; Need ultrasonic)
Grade Clinical information: Phase 1
Molecular Formula C20H17F2N3O3
Molecular Weight 385.36
CAS-Number [1464842-09-8]
Storage Conditions Please store the product under the recommended conditions in the Certificate of Analysis.
Product Line Research
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Material Safety Data Sheet Download PDF
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