GPR81 agonist 1


Catalog Number Pack Size List Price* Quantity
HY-135982-5MG 5 mg 521,00 Add
HY-135982-1ML 10mM/1mL 571,00 Add
HY-135982-10MG 10 mg 875,00 Add
HY-135982-50MG 50 mg 2'484,00 Add
HY-135982-100MG 100 mg 3'687,00 Add

* CHF, excl. 8.1% VAT and shipping costs


Product Description

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GPR81 agonist 1 is a potent and highly selective GPR81 agonist, with EC50s of 58 nM and 50 nM for human and mouse GPR81, respectively. GPR81 agonist 1 inhibits lipolysis in differentiated 3T3-L1 adipocytes. GPR81 agonist 1 suppresses lipolysis in mice without cutaneous flushing. GPR81 agonist 1 displays remarkable selectivity for GPR81 over GPR109a[1].

Category Biochemicals
Supplier MedChem Express
Regulatory Status RUO
Research Field Metabolic Disease, GPCR/G Protein
Format Solubility: DMSO : 50 mg/mL (ultrasonic)
Grade Clinical information: No Development Reported
Purity 99.78%
Molecular Formula C22H30N4O2S2
Molecular Weight 446.63
CAS-Number 1620992-67-7
Storage Conditions -20°C, 3 years; 4°C, 2 years (Powder)
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Shipping Details Room Temperature
Material Safety Data Sheet Download PDF