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GPR81 agonist 1


Catalog Number Pack Size List Price* Quantity
HY-135982-50MG 50 mg Inquire
HY-135982-5MG 5 mg Inquire
HY-135982-10MG 10 mg Inquire
HY-135982-100MG 100 mg Inquire

* CHF, excl. 7.7% VAT and shipping costs


Product Description

GPR81 agonist 1 is a potent and highly selective GPR81 agonist, with EC50s of 58 nM and 50 nM for human and mouse GPR81, respectively. GPR81 agonist 1 inhibits lipolysis in differentiated 3T3-L1 adipocytes. GPR81 agonist 1 suppresses lipolysis in mice without cutaneous flushing. GPR81 agonist 1 displays remarkable selectivity for GPR81 over GPR109a.

Category Biochemicals
Supplier MedChem Express
Application Metabolism-protein/nucleotide metabolism
Regulatory Status RUO
Grade Clinical information: No Development Reported
Molecular Formula C22H30N4O2S2
Molecular Weight 446.63
CAS-Number [1620992-67-7]
Storage Conditions Please store the product under the recommended conditions in the Certificate of Analysis.
Product Line Research
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Material Safety Data Sheet Download PDF
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