Logo Lucerna-Chem
+41 41 420 9636

Regulatory Status

Article Status


Catalog Number Pack Size List Price* Quantity
HY-18618-5MG 5 mg Inquire
HY-18618-10MG 10 mg Inquire

* CHF, excl. 7.7% VAT and shipping costs

Product Description

SB-612111 is a novel and potent opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model.

Category Biochemicals
Supplier MedChem Express
Application COVID-19-immunoregulation
Regulatory Status RUO
Grade Clinical information: No Development Reported
Molecular Formula C24H29Cl2NO
Molecular Weight 418.4
CAS-Number [371980-98-2]
Storage Conditions Please store the product under the recommended conditions in the Certificate of Analysis.
Product Line Research
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Material Safety Data Sheet Download PDF
Call us

Customer Support
T +41 41 420 96 36
F +41 41 420 96 56

Business Hours
From Monday through Friday
08:00 – 12:00
13:00 – 17:00

Ask us

Technical Support

Business Development

Postal address
Lucerna-Chem AG
Abendweg 18
CH-6006 Luzern


If you have already subscribed to our newsletter and would like to update your details or cancel it, please click here.

© Copyright 2021 Lucerna-Chem AG, Switzerland