SB-612111
Catalog Number | Pack Size | List Price* | Quantity | |
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HY-18618-1ST | Get quote | Inquire |
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Product Description
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SB-612111 is a novel and potent opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1].
Category | Biochemicals |
Supplier | MedChem Express |
Regulatory Status | RUO |
Research Field | Inflammation/Immunology, Neurological Disease, GPCR/G Protein,Neuronal Signaling |
Format | Solubility: 10 mM in DMSO |
Grade | Clinical information: No Development Reported |
Molecular Formula | C24H29Cl2NO |
Molecular Weight | 418.4 |
CAS-Number | 371980-98-2 |
Tech. Data Sheet | View datasheet |
Link To Supplier | http://www.medchemexpress.com |
Shipping Details | Room temperature |
Material Safety Data Sheet | Download PDF |