GSK8814
| Catalog Number | Pack Size | List Price* | Quantity | |
|---|---|---|---|---|
| HY-114204-5MG | 5 mg | 597,00 | Add | |
| HY-114204-1ML | 10mM/1mL | 655,00 | Add | |
| HY-114204-10MG | 10 mg | 1'001,00 | Add |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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GSK8814 is a potent, selective, and ATAD2/2B bromodomain chemical probe and inhibitor, with a binding constant pKd=8.1 and a pKi=8.9 in BROMOscan. GSK8814 binds to ATAD2 and BRD4 BD1 with pIC50s of 7.3 and 4.6, respectively. GSK8814 shows 500-fold selectivity for ATAD2 over BRD4 BD1[1].
| Category | Biochemicals |
| Supplier | MedChem Express |
| Regulatory Status | RUO |
| Research Field | Cancer, Epigenetics |
| Format | Solubility: DMSO : 100 mg/mL (ultrasonic) |
| Grade | Clinical information: No Development Reported |
| Purity | 99.6% |
| Molecular Formula | C28H35F2N5O3 |
| Molecular Weight | 527.61 |
| CAS-Number | 1997369-78-4 |
| Storage Conditions | -20°C, 3 years (Powder) |
| Tech. Data Sheet | View datasheet |
| Link To Supplier | http://www.medchemexpress.com |
| Shipping Details | Blue Ice |
| Material Safety Data Sheet | Download PDF |
